PerkinElmer

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二元彩票网 www.mwbxj.com

Simplify the development of your assays and the calculation of your results using our radioligands, receptor-transfected cell membranes, and cell lines for radioligand binding applications.

Because radioligands can be directly detected, there is no need to generate intermediate antibodies against your target. Eliminating these antibodies also eliminates the need to optimize an antibody titer and reduces your total assay time by skipping intermediate incubation steps.

You’ll find our receptor-ligand binding reagents and related products perfect matches for all of your receptor binding studies.

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"受体配体结合" 1-50530 产品与服务

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UNIFILTER-24 孔细胞收集器

速度快、操作简单是Unifilter收集器的主要优势。

OMNIFILTER-96 孔细胞收集器

速度快、操作简单是OmniFilter收集器的主要优势。

MICROBETA FILTERMAT-24 孔细胞收集器

速度快、操作简单是 Filtermate 收集器的主要优势。FilterMate 系统的整个操作过程都很简便。若需要更多信息,请点击产品上的选项卡。

UNIFILTER-96 孔细胞收集器 SS

速度快、操作简单是Unifilter收集器的主要优势。

MICROBETA FILTERMAT-96 孔细胞收集器

速度快、操作简单是 Filtermate 收集器的主要优势。FilterMate 系统的整个操作过程都很简便。

UNIFILTER-96 孔细胞收集器

速度快、操作简单是Unifilter收集器的主要优势。
LabChip EZ Reader

酶动力学读板仪

酶动力学读板仪以更低的时间和经费成本,帮您的实验室更快的发现最有潜力的候选化合物。
Receptor-expressing cell lines

ValiScreen Adrenergic alpha 2A (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

WGA PVT SPA 100 MG

WGA-coated SPA beads, for capturing cell membranes in proximity-based radiometric scintillation assays.

Bradykinin, [2,3-Prolyl-3,4-3H(N)]

Bradykinin, tritiated at the 2,3-prolyl-3,4 position. Bradykinin is the endogenous ligand that activates bradykinin B1 and B2 receptors.
Receptor-expressing cell lines

ValiScreen Neuropeptide Y Y2 (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

p53 Acetylated Peptide, for LabChip EZ Reader

Fluorescently-labelled p53 Peptide (Acetylated) for Epigenetic Assays (Enzyme inhibiton, target discovery, lead optimization)
PerkinElmer

Membrane Target Systems: Bombesin BB2 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
PerkinElmer

Membrane Target Systems: GABA B1a (human) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from CHO-K1 cells stably-transfected with human GABA B1a receptor, 400 units.

NALOXONE, [N-ALLYL-2,3-3H]-

Naloxone radioligand tritiated at the 2,3 position. Naloxone acts as a non-selective, competitive opioid receptor antagonist.

Vinblastine Sulphate, [G-3H]

Vinblastine sulphate, tritiated. Vinblastine binds to tubulin and inhibits microtubule formation.

Citalopram, [N-Methyl-3H]

Citalopram, tritiated at the N-methyl group. Citalopram is a selective serotonin reuptake inhibitor (SSRI) antidpressant drug, and has been shown to block the serotonin transporter (SERT, 5-HTT).

MESULERGINE, [N-METHYL-3H]-, 250 μCi

Mesulergine, tritiated on the N-methyl group. Mesulergine acts as an antagonist at serotonin 5-HT2A and 5-HT2C receptors, and as a partial agonist at dopamine receptors.
PerkinElmer

ProfilerPro Kinase Selectivity Assay Plate Kit 4, for LabChip EZ Reader

Kit consist of matched pairs of 384-well kinase-assay and substrate plates. Each assay plate contains 24 different predispensed frozen kinases. Substrate plates contain the appropriate fluorescent labeled peptides and ATP.
Receptor-expressing cell lines

ValiScreen Prostanoid DP (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Membrane Target Systems: Adrenergic alpha 1A (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.

Verapamil Hydrochloride, [N-Methyl-3H]

Verapamil hydrochloride, tritiated on the N-methyl group. Verapamil acts as a calcium channel blocker (CCB).

Glibenclamide, Glyburide, [Cyclohexyl-2,3-3H(N)]-, 250μCi (9.25MBq)

Glibenclamide (glyburide) tritiated at the cyclohexyl-2,3 position. Glibenclamide is an antidiabetic drug that binds and inhibits the ATP-sensitive potassium channel.
Receptor-expressing cell lines

ValiScreen Vasopressin V1b (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Neurokinin B, [125I]His, MePhe7

Neurokinin B (NKB), labeled with 125I on the histidine residue. Neurokinin B is involved in ovarian cycle regulation, and binds neurokinin 3 receptor (NK3R; tachykinin receptor 3), a GPCR involved in vascular remodeling, angiogenesis, and cancer.
Receptor-expressing cell lines

ValiScreen N-formyl Peptide (FPRL1) (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.
PerkinElmer

Streptavidin PVT 500MG

Streptavidin-coated SPA beads, for capturing biotinylated biomolecules in proximity-based radiometric scintillation assays.
PerkinElmer

Membrane Target Systems: Galanin Gal1 (human) membrane preparation, in HEK-293 cells. 400 Units.

Cell membranes prepared from HEK293 cells stably-transfected with human galanin Gal1 receptor, 400 units.
PerkinElmer

Membrane Target Systems: Chemoattractant C5a (human varient) membrane preparation, in CHO-K1 cells. 400 Units.

Cell membranes prepared from CHO-K1 cells stably-transfected with human chemoattractant C5a (human varient) receptor, 400 units.

(-)-CGP-12177, [5,7-3H]

(-)-CGP-12177 radioligand tritiated at the 5,7 position. CGP-12177 acts as an antagonist at the β1- and β2-adrenoceptors and a partial agonist at β3-adrenoceptors.

Histamine Dihydrochloride, [Ring, Methylenes-3H(N)]

Histamine dihydrochloride, tritiated on the ring and methylene groups. Histamine is an endogenous agonist of histamine receptors.
PerkinElmer

Membrane Target Systems: Neuromedin U NMU1 (FM3) (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.
PerkinElmer

Membrane Target Systems: Calcitonin CGRP1 (human) membrane preparation, in CHO-K1 cells. 400 Units.

Our Membrane Target System membranes are prepared from cells that express recombinant or endogenous receptors. Selected for optimal performance in binding assays.

Orexin A, [125I]

Orexin A, labeled with 125I. Orexin A binds to orexin receptors (OX1 and OX2), which are potential drug targets for sleep disorders.
PerkinElmer

Histone 4 Acetylated Peptide, for LabChip EZ Reader

Fluorescently-labelled Histone 4 Peptide (Acetylated) for Epigenetic Assays (Enzyme inhibiton, target discovery, lead optimization)

Ω-Conotoxin MVIIC, [125I]

Ω-Conotoxin MVIIC (ω-Conotoxin MVIIC), labeled with 125I. Ω-Conotoxin MVIIC is a neurotoxin that blocks calcium channels.
PerkinElmer

ProfilerPro Kinase Selectivity Assay Plate Kit 3, for LabChip EZ Reader

Kit consist of matched pairs of 384-well kinase-assay and substrate plates. Each assay plate contains 24 different predispensed frozen kinases. Substrate plates contain the appropriate fluorescent labeled peptides and ATP.

2-Methylthio ADP, [β-33P]-, 10mM Tricine (pH 7.6)

33P labeled 2-methyl-thio ADP (2-MeS-ADP), labeled on the beta phosphate group. 2-MeS-ADP acts as an agonist at P2Y1, P2Y12, and P2Y13 receptors and is used in platelet aggregation research.

Substance-P (9-Sar, 11-Met(O2)), [2-Prolyl-3,4-3H]-, 50μCi (1.85MBq)

Substance-P, tritiated on the 2-prolyl group. Substance-P acts as an antagonist at neurokinin-1 receptors (NK1Rs).
PerkinElmer

PEI PS Imaging Beads 50 MG

SPA imaging beads coated with polyethyleneimine (PEI) to decrease non-specific binding. These beads are commonly used in receptor binding assays.
PerkinElmer

Streptavidin YSI 75MG

Streptavidin-coated SPA beads, for capturing biotinylated biomolecules in proximity-based radiometric scintillation assays.
Receptor-expressing cell lines

ValiScreen Chemotactic Peptide C3a (human) cell line

Our stable recombinant ValiScreen cell lines express a variety of GPCRs for binding and functional assays.

Vasopressin (8-L-Arginine), [Phenylalanyl-3,4,5-3H(N)]

Vasopressin, tritiated on the phenylalanine residue. Vasopressin binds and activates vasopressin receptors.
PerkinElmer

ProfilerPro Kinase Peptide Substrate 1, for LabChip EZ Reader

Fluorescently-labelled peptide substrate 1 for kinase assays (inhibiton, target discovery, lead optimization)

Somatostatin, [125I]Tyr11

Somatostatin, labeled with 125I. Somatostatin binds somatostatin receptors, and inhibits the secretion of insulin and glucagon.

INSULIN (porcine), [125I], 10μCi (370kBq), Specific Activity:80-120μCi (2.96-4.44MBq)/μg

Insulin (porcine), labeled with 125I. Insulin is a peptide hormone that binds to insulin receptors to increase cellular uptake of glucose, increase DNA replication and protein synthesis, and modify enzymatic activity. This product is radioiodinated with 125I using a modification of the Hunter and Greenwood method and purified by ion-exchange column chromatography. This method predominantly labels tyrosine residues.
PerkinElmer

WGA YSI 1G

WGA-coated SPA beads, for capturing cell membranes in proximity-based radiometric scintillation assays.

Ornithine Vasotocin Analog, [125I]-OVTA)

Ornithine Vasotocin Analog (OVTA), labeled with 125I. OVTA binds oxytocin receptors, a hormone receptor involved in pregnancy, milk production, stress, social memory, and bonding.

Iodo-Melatonin, 2-[125I]

Melatonin, labeled with 125I. Melatonin binds and activates melatonin receptors, a class of GPCRs that are potential drug targets for circadian rhythm sleep disorders and depression.

"受体配体结合" 1-50530 产品与服务

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